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After 1 year, 47.5% of the patients in the lorcaserin group and 20.3% in the placebo group had lost 5% or more of their body weight

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Under identical conditions, treatment with PF-06882961 led to FAP-GLP-1R internalization (EC 50 = 230 nM, E max = 83%)

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Instead, the focus should be on reducing avoidable triggers for shedding

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